Inhibitors - Page 511

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Biological type of action

Agonists(items: 859)

Inhibitors(items: 13224)

Inhibitors

Pfizer compound category

Compounds with inhibitory activity towards a wide range of targets

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EBC-220134
EBC-220134

CAS:1372540-25-4

2-methyl-1-{[2-methyl-3-(trifluoromethyl)phenyl]methyl}-6-(morpholin-4-yl)-1H-1,3-benzodiazole-4-carboxylic acid
2-methyl-1-{[2-methy...
-

1

+
EBC-220140
EBC-220140

CAS:2049868-46-2

2,2-dimethyl-1-[(5S)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl]propan-1-one
2,2-dimethyl-1-[(5S)...
-

1

+
EBC-220143
EBC-220143

CAS:220904-83-6

GW 5074
GW 5074
-

1

+
EBC-220145
EBC-220145

CAS:1457983-28-6

G749
G749
-

1

+
EBC-220148
EBC-220148

CAS:1075200-91-7

N-{2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1H-indol-5-yl}ethane-1-sulfonamide
N-{2-oxo-3-[phenyl({...
-

1

+
EBC-220150
EBC-220150

CAS:1702259-66-2

N-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}prop-2-enamide
N-{2-[(6-{[(2,6-dich...
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1

+
EBC-220178
EBC-220178

CAS:1800398-38-2

N-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide
N-{3-[2-(2-hydroxyet...
-

1

+
EBC-220181
EBC-220181

CAS:871357-89-0

(1S,2S,3R,4R)-3-[(5-fluoro-2-{[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide
(1S,2S,3R,4R)-3-[(5-...
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1

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EBC-220189
EBC-220189

CAS:

4-fluoro-N-(6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[(1s,4s)-4-[(propan-2-yl)carbamoyl]cyclohexyl]-1H-1,3-benzodiazol-2-yl)benzamide
4-fluoro-N-(6-{[4-(2...
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1

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EBC-220193
EBC-220193

CAS:866405-64-3

4-(6-{4-[2-(piperidin-1-yl)ethoxy]phenyl}pyrazolo[1,5-a]pyrimidin-3-yl)pyridine
4-(6-{4-[2-(piperidi...
-

1

+
EBC-220198
EBC-220198

CAS:1257628-77-5

Olverembatinib
Olverembatinib
-

1

+
EBC-221024
EBC-221024

CAS:545-47-1

Lupeol
Lupeol
-

1

+
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