Inhibitors - Page 510

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Biological type of action

Agonists(items: 859)

Inhibitors(items: 13224)

Inhibitors

Pfizer compound category

Compounds with inhibitory activity towards a wide range of targets

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EBC-220039
EBC-220039

CAS:944396-07-0

Buparlisib
Buparlisib
-

1

+
EBC-220040
EBC-220040

CAS:

3-{3-[({4-[(dimethylamino)methyl]phenyl}amino)(phenyl)methylidene]-2-oxo-2,3-dihydro-1H-indol-6-yl}-N-ethylprop-2-ynamide
3-{3-[({4-[(dimethyl...
-

1

+
EBC-220046
EBC-220046

CAS:1001350-96-4

(2S)-1-{4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}-N-(6-fluoropyridin-3-yl)-2-methylpyrrolidine-2-carboxamide
(2S)-1-{4-[(5-cyclop...
-

1

+
EBC-220048
EBC-220048

CAS:

7-(2-hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide
7-(2-hydroxypropan-2...
-

1

+
EBC-220050
EBC-220050

CAS:649735-46-6

Brivanib
Brivanib
-

1

+
EBC-220052
EBC-220052

CAS:

N-{3-[(5-bromo-4-{[2-(1H-imidazol-5-yl)ethyl]amino}pyrimidin-2-yl)amino]phenyl}pyrrolidine-1-carboxamide
N-{3-[(5-bromo-4-{[2...
-

1

+
EBC-220057
EBC-220057

CAS:

1-[4-(6-bromo-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-3H-imidazo[4,5-b]pyridin-2-yl)phenyl]-4-methylpiperazine
1-[4-(6-bromo-7-{4-[...
-

1

+
EBC-220062
EBC-220062

CAS:1202757-89-8

AVL-292
AVL-292
-

1

+
EBC-220075
EBC-220075

CAS:1265229-25-1

Zoligratinib
Zoligratinib
-

1

+
EBC-220112
EBC-220112

CAS:1382979-44-3

5-[6,6-dimethyl-4-(morpholin-4-yl)-6H,8H,9H-[1,4]oxazino[3,4-h]purin-2-yl]pyrimidin-2-amine
5-[6,6-dimethyl-4-(m...
-

1

+
EBC-220120
EBC-220120

CAS:778270-11-4

3-(6-{[4-(trifluoromethoxy)phenyl]amino}pyrimidin-4-yl)benzamide
3-(6-{[4-(trifluorom...
-

1

+
EBC-220125
EBC-220125

CAS:958852-01-2

GSK1059615
GSK1059615
-

1

+
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