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EBCL-0045

Bioactive Compounds Max

The Library of Bioactive Compounds Max is our most extensive collection, featuring 14388 compounds with known biological activity, including a diverse range of drug candidates, tool compounds, metabolites, prodrugs, and approved drugs.

Each compound is fully annotated with detailed biological activity data and supported by literature references, ensuring comprehensive and up-to-date information.We also offer custom synthesis and compound sourcing, allowing access to nearly any compound through our in-house capabilities, making this library an invaluable resource for drug discovery, repurposing, and research applications.

Related Terms: bioactivity, biological targeting, GPCR, carbonic anhydrase, ligand-gated ion channel.

Preplated options

Dry powder/solution (DMSO)Dry powder
Number of compounds12386
Comment
Dry powder/solution (DMSO)DMSO
Number of compounds10270
Comment

Highlights

Molecule highlight
EBC-65074CAS: 1007648-66-9

This compound is an inhibitor of Farnesoid X receptor.

Molecule highlight
EBC-08969CAS: 941032-88-8

This compound is an inhibitor of poly polymerase 1.

Molecule highlight
EBC-157131CAS: 351424-20-9

CBA is a potent and selective inhibitor of the cation channel TRPM4, with an IC50 of 1.1 μM.

Molecule highlight
EBC-291143CAS: 338989-14-3

This compound inhibits acetylcholinesterase and carbonic anhydrases CA II and CA I.

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Disclaimer

All our products are for research purpose only. Any personal or non-scientific use is strictly prohibited.

Note

All the compounds with solubility below 10 mM are shipped as 2 mM solutions.

Product Features

Library of Bioactive Compounds Max is a set of 14388 bioactive molecules for HTS/HCS programs.

The Library of Bioactive Compounds Max covers novel promising preclinical lead compounds, clinical candidates and approved drugs.

Calculated structural diversity of the collection: 0.87.

Comprehensive documentation with structures, trivial names, synonyms, activity coefficient values, types of action on target and references to original literature.

NMR and LCMS validated purity.All the compounds are available in stock for hit follow-up.

The library is continuously updated.

Product Details

  • Format: 10 - 100 µL of 10 mM DMSO stock solutions; dry powders (1 mg);
  • Container: 384-well microplates;
  • Storage: - 18 °C;
  • Shipping: Dry ice.

Utility

  • High throughput screening (HTS);
  • High content screening (HCS);
  • Cherry picking.