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EBCL-0003

Bioactive Compounds III

Bioactive Library III is a collection of 1703 compounds with annotated biological activity. This collection is based on Bioactive Library I and contains compounds with sub-ten nanomolar activity coefficient values only.

  • Fully annotated: all compounds are provided with literature references and detailed and up to date biological activity data.
  • Custom Synthesis and Compound Sourcing: we can supply almost any compound either via in-house synthesis or using our supplier network.


Related terms:  carbonic anhydrase, D2 receptor, H1 receptor, 5-HT2A, fatty acid amide hydrolase, D3, epidermal growth factor, SERT, acetylcholinesterase

Library image center

Preplated options

Dry powder/solution (DMSO)Dry powder
Number of compounds1703
Comment
Dry powder/solution (DMSO)DMSO
Number of compounds1454
Comment

Highlights

Molecule highlight
EBC-11162CAS: 41340-25-4

Etodolac is a non-steroidal anti-inflammatory drug (NSAID). It is indicated for relief of signs and symptoms of rheumatoid arthritis and osteoarthritis.

Molecule highlight
EBC-06639CAS: 66611-26-5

RU 24969 is a 5-hydroxytryptamine receptor 1b inhibitor with Ki (inhibition constant) = 0.43 nM

Molecule highlight
EBC-03656CAS: 2736-23-4

2,4-Dichloro-5-sulfamoylbenzoic acid is a carbonic anhydrase inhibitor with Kd (dissociation constant) = 0.14 nM

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Disclaimer

All our products are for research purpose only. Any personal or non-scientific use is strictly prohibited.

Note

All the compounds with solubility below 10 mM are shipped as 2 mM solutions.

Product Features

  • Enamine Bioactive Library III is a set of 1703 bioactive molecules for HTS/HCS programs.
  • The Bioactive Library III covers novel promising preclinical lead compounds, clinical candidates and approved drugs.
  • Comprehensive documentation with structures, trivial names, synonyms, activity coefficient values, types of action on target and references to original literature.
  • NMR and LCMS validated purity.
  • All the compounds are available in stock for hit follow-up.
  • The library is continuously updated.

Product Details

  • Format: 10 - 100 µL of 10 mM DMSO stock solutions; dry powders (1 mg);
  • Container: 384-well microplates;
  • Storage: - 18 °C;
  • Shipping: Dry ice.

Utility

  • High throughput screening (HTS);
  • High content screening (HCS);
  • Cherry picking.

Library Composition

Name
Occurrence in the library, times

carbonic anhydrase 2

50

50

Number of compounds

50

carbonic anhydrase 12

36

36

Number of compounds

36

D2 receptor

33

33

Number of compounds

33

H1 receptor

33

33

Number of compounds

33

5-HT2A receptor

32

32

Number of compounds

32

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