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Product details:
ID
CAS
1672662-14-4
Purity
95%
PT2399 is a potent and selective EPAS1 antagonist, which directly binds to EPAS1 PAS B domain with an IC50 of 6 nM. PT2399 displays potent antitumor activity in vivo.
Properties
Name
PT2399
Smiles
O[C@H]1C=2C(CC1(F)F)=C(OC=3C=C(F)C=C(C#N)C3)C=CC2S(=O)(=O)C(F)F
Targets
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Target name
Target pX
Target action
doi
SDS
PT2399
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$150
2 mg
$150
5 mg
$228
10 mg
$394
15 mg
$477
20 mg
$560
25 mg
$682
30 mg
$803
35 mg
$924
40 mg
$1045
45 mg
$1120
50 mg
$1196
75 mg
$1590
100 mg
$POA
Quantity
1
Total amount
$ 228
PT2399
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.