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Product details:
CAS
149838-21-1
Purity
95%
PD-85639 is a voltage-gated sodium (Na+) channel blocker that is shown to target rat brain Nav1.2 with simultaneous high- and low-affinity modes of binding and a fast kinetic, competitive against the local anesthetic Na+ channel blockers tetracaine, bupivacaine, and mepivacaine, as well as Na+ channel activators veratridine and batrachotoxin.
Properties
Name
PD-85639
Smiles
CC1CCCC(C)N1CCCNC(=O)C(C=2C=CC=CC2)C=3C=CC=CC3
Targets
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Sold for research purposes under agreement from Pfizer Inc.
SDS
PD 85639 | [3H]-PD 85639
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$94
2 mg
$98
5 mg
$102
10 mg
$122
15 mg
$165
20 mg
$208
25 mg
$247
30 mg
$288
35 mg
$319
40 mg
$351
45 mg
$378
50 mg
$417
75 mg
$576
100 mg
$POA
Quantity
1
Total amount
$ 102
PD 85639 | [3H]-PD 85639
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.