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Product details:

SPH3127

Search by this structure
Molecule product

ID

EBC-420057

CAS

1399849-02-5

Purity

95%

SPH3127 appears to be a very potent DRI with much improved PK properties compared to the earlier compounds. It potently inhibits REN with an IC50 = 0.4 nM.

Properties

cLogP:1.001
MW:444.527

Name

SPH3127

Smiles

COC(=O)NCCCN1N=C([C@@H](C)N(C2CC2)C(=O)[C@H]3CNCCO3)C=4C=CC(C)=NC14

Targets

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Chemical probes

Target name

Target pX

Target action

doi

Renin

9.4

Inhibitor

Open link
Synonyms

SPH3127

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Prices

Temporarily unavailable

1 mg

$210

2 mg

$315

5 mg

$629

10 mg

$1090

15 mg

$1320

20 mg

$1550

25 mg

$1886

30 mg

$2221

35 mg

$2556

40 mg

$2891

45 mg

$3100

50 mg

$3310

75 mg

$4399

100 mg

$POA

Quantity

-

1

+

Total amount

$ 629

Your current project

Temporarily unavailable

Synonyms

SPH3127

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Target activity features

It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.

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