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Product details:

PF-04995274

Molecule product

ID

EBC-384061

|

PF-04995274

CAS

1331782-27-4

Purity

95%

PF-04995274 is a partial agonist of the 5-hydroxytryptamine receptor subtypes 5-HT4A, 5-HT4B, 5-HT4D, and 5-HT4E with Ki values of 0.36, 0.46, 0.33, and 0.32 nM, respectively, in a radioligand binding assay.

Properties

cLogP:1.684
MW:432.51

Name

PF-04995274

Smiles

OC1(CN2CCC(COC3=NOC=4C=CC=C(O[C@@H]5CCOC5)C34)CC2)CCOCC1

Targets

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Licensing Information

Sold for research purposes under agreement from Pfizer Inc.

Product datasheets

SDS

Synonyms

PF-04995274

Transportation & Handlings
Storage temperature:+4
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Molarity Calculator
Dilution Calculator
Formulation Calculator

Prices

1 mg

$85

2 mg

$85

5 mg

$85

10 mg

$92

15 mg

$111

20 mg

$131

25 mg

$159

30 mg

$187

35 mg

$215

40 mg

$244

45 mg

$261

50 mg

$278

75 mg

$371

100 mg

$POA

Quantity

-

1

+

Total amount

$ 85

Your current project

In Stock

Synonyms

PF-04995274

Transportation & Handlings
Storage temperature:+4
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Target activity features

It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.