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CAS
66504-75-4
Purity
95%
Bicifadine hydrochloride is a potent antagonist of SLC6A2 (noradrenalin transporter) (IC50 = 54.7 nM). Bicifadine also has antagonistic activity at the 5-HT receptors and dopamine transporters (IC50 = 117 nM and 910 nM, respectively). It exhibits antinociceptive and antiallodynic properties in rodent models of acute, persistent, and chronic pain.
Properties
Name
Bicifadine hydrochloride
Smiles
Cl.CC=1C=CC(=CC1)C23CC3CNC2
Targets
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(+)-1-(p-tolyl)-3-azabicyclo[3.1.0]hexane hydrochloride | 1-(4-methylphenyl)-3-azabicyclo hexane hydrochloride | 1-(4-methylphenyl)-3-azabicyclo[3.1.0]hexane hydrochloride | Bicifadine hydrochloride | bicifadine
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$67
2 mg
$71
5 mg
$78
10 mg
$102
15 mg
$116
20 mg
$129
25 mg
$141
30 mg
$149
35 mg
$164
40 mg
$182
45 mg
$194
50 mg
$208
75 mg
$300
100 mg
$344
Quantity
1
Total amount
$ 78
(+)-1-(p-tolyl)-3-azabicyclo[3.1.0]hexane hydrochloride | 1-(4-methylphenyl)-3-azabicyclo hexane hydrochloride | 1-(4-methylphenyl)-3-azabicyclo[3.1.0]hexane hydrochloride | Bicifadine hydrochloride | bicifadine
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.
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