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Product details:

Phentolamine mesylate

Molecule product

ID

EBC-153121

CAS

65-28-1

Purity

95%

Phentolamine produces its therapeutic actions by competitively blocking alpha-adrenergic receptors, leading to a muscle relaxation and a widening of the blood vessels. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, vasospasm of raynaud disease and frostbite, clonidine withdrawal syndrome, impotence, and peripheral vascular disease.

Properties

cLogP:3.809
MW:377.141

Name

Phentolamine mesylate

Smiles

CC=1C=CC(=CC1)N(CC2=NCCN2)C=3C=CC=C(O)C3.CS(=O)(=O)O

Targets

Please log in to see this information

Product datasheets

SDS

Synonyms

phentolamine mesylate

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Molarity Calculator
Dilution Calculator
Formulation Calculator

Prices

1 mg

$19

2 mg

$19

5 mg

$19

10 mg

$19

15 mg

$19

20 mg

$19

25 mg

$19

30 mg

$19

35 mg

$19

40 mg

$19

45 mg

$19

50 mg

$19

75 mg

$19

100 mg

$POA

Quantity

-

1

+

Total amount

$ 19

Your current project

In Stock

Synonyms

phentolamine mesylate

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Target activity features

It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.

Related Compounds

EBC-15029
EBC-15029

CAS:249607-96-3

3-{[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino}phenol; acetic acid
3-{[(4,5-dihydro-1H-...
-

0

+
EBC-478105
EBC-478105

CAS:

3-{[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino}(4-2H)phenol
3-{[(4,5-dihydro-1H-...
-

0

+
EBC-26433
EBC-26433

CAS:50-60-2

3-{[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino}phenol
3-{[(4,5-dihydro-1H-...
-

0

+