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Product details:
CAS
1884640-99-6
Purity
95%
NI-42 is a new chemical probe for the BRPFs (bromodomain and PHD finger-containing). It is a potent inhibitor of the BRD of the BRPFs with IC50s of 7.9, 48, 260 nM for BRPF1, BRPF2, BRPF3.
Properties
Name
NI-42
Smiles
CC1=CC=2C=C(NS(=O)(=O)C=3C=CC(C#N)=CC3)C=CC2N(C)C1=O
Targets
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Sold for research purposes under agreement from Pfizer Inc.
SDS
No records
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$56
2 mg
$61
5 mg
$66
10 mg
$83
15 mg
$91
20 mg
$99
25 mg
$111
30 mg
$118
35 mg
$127
40 mg
$143
45 mg
$153
50 mg
$165
75 mg
$235
100 mg
$POA
Quantity
1
Total amount
$ 66
No records
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.
