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Product details:

Lapatanib

Molecule product

ID

EBC-00694

CAS

231277-92-2

Purity

95%

Lapatinib is a 4-anilinoquinazoline kinase inhibitor of the intracellular tyrosine kinase domains of both epidermal growth factor receptor (HER1/EGFR/ERBB1) and human epidermal growth factor receptor type 2 (HER2/ERBB2). Lapatinib is an anti-cancer drug, used for the treatment for solid tumours such as breast and lung cancer.

Properties

cLogP:5.965
MW:581.058
Pharmacopoeia:FDA

Name

Lapatanib

Smiles

CS(=O)(=O)CCNCC1=CC=C(O1)C=2C=CC=3N=CN=C(NC=4C=CC(OCC=5C=CC=C(F)C5)=C(Cl)C4)C3C2

Targets

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Product datasheets

SDS

Synonyms

GW-572016 | LAP | Lapatinib | apatinib | lapatanib | tykerb | tyverb

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility
Solvent
Measure
Concentration
Unit
DMSO
215.12
uM
DMSO
10
Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Molarity Calculator
Dilution Calculator
Formulation Calculator

Prices

1 mg

$19

2 mg

$19

5 mg

$19

10 mg

$19

15 mg

$19

20 mg

$19

25 mg

$19

30 mg

$19

35 mg

$19

40 mg

$19

45 mg

$19

50 mg

$19

75 mg

$19

100 mg

$POA

Quantity

-

1

+

Total amount

$ 19

Your current project

In Stock

Synonyms

GW-572016 | LAP | Lapatinib | apatinib | lapatanib | tykerb | tyverb

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility
Solvent
Measure
Concentration
Unit
DMSO
215.12
uM
DMSO
10
Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Target activity features

It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.

Related Compounds

EBC-08811
EBC-08811

CAS:388082-78-8

bis(4-methylbenzene-1-sulfonic acid); N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(5-{[(2-methanesulfonylethyl)amino]methyl}furan-2-yl)quinazolin-4-amine
bis(4-methylbenzene-...
-

0

+
EBC-35022
EBC-35022

CAS:1187538-35-7

4-methylbenzene-1-sulfonic acid; N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(5-{[(2-methanesulfonylethyl)amino]methyl}furan-2-yl)quinazolin-4-amine
4-methylbenzene-1-su...
-

0

+
EBC-00694
EBC-00694

CAS:231277-92-2

N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(5-{[(2-methanesulfonylethyl)amino]methyl}furan-2-yl)quinazolin-4-amine
N-{3-chloro-4-[(3-fl...
-

0

+