Inhibitors - Page 783

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Biological type of action

Agonists(items: 859)

Inhibitors(items: 13223)

Inhibitors

Pfizer compound category

Compounds with inhibitory activity towards a wide range of targets

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EBC-608280
EBC-608280

CAS:916173-19-8

2-{1H-pyrrolo[2,3-b]pyridin-4-yl}aniline
2-{1H-pyrrolo[2,3-b]...
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1

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EBC-608281
EBC-608281

CAS:20320-52-9

2-[2-(dimethylamino)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(dimethylamino)...
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1

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EBC-608309
EBC-608309

CAS:904504-22-9

5-hydroxy-16,17-dimethoxy-1,11-diazapentacyclo[10.7.1.0^{2,7}.0^{8,20}.0^{13,18}]icosa-2(7),3,5,8,10,12(20),13(18),14,16-nonaen-19-one
5-hydroxy-16,17-dime...
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1

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EBC-608311
EBC-608311

CAS:58722-34-2

1-[4-(piperidine-1-sulfonyl)phenyl]ethan-1-one
1-[4-(piperidine-1-s...
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1

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EBC-609077
EBC-609077

CAS:2270189-42-7

6-[(dimethylamino)methyl]-5-iodo-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-[(dimethylamino)me...
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1

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EBC-609078
EBC-609078

CAS:2715287-71-9

5-[4-(morpholin-4-yl)-6-(piperazin-1-yl)-1,3,5-triazin-2-yl]-1,3-benzoxazol-2-amine
5-[4-(morpholin-4-yl...
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1

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EBC-609080
EBC-609080

CAS:682745-59-1

(2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-methoxyphenyl)methyl]sulfanyl}-9H-purin-9-yl)oxolane-3,4-diol
(2R,3S,4R,5R)-2-(hyd...
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1

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EBC-609082
EBC-609082

CAS:2244129-20-0

3-(isoquinolin-8-yloxy)-4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(4-methylpiperazin-1-yl)phenyl]benzamide
3-(isoquinolin-8-ylo...
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1

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EBC-609083
EBC-609083

CAS:1400941-89-0

N-[(3-{[(2-amino-9H-purin-6-yl)oxy]methyl}phenyl)methyl]acetamide
N-[(3-{[(2-amino-9H-...
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1

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EBC-609084
EBC-609084

CAS:

3-chloro-N'-[(E)-(3,5-dimethoxy-4-{[4-(propan-2-yl)phenyl]methoxy}phenyl)methylidene]-4-hydroxybenzohydrazide
3-chloro-N'-[(E)-(3,...
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1

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EBC-609085
EBC-609085

CAS:

(1S,2S,3R,4R)-3-{[5-(5-fluoropyridin-3-yl)-2-{[3-(pyrrolidine-1-carbonyl)phenyl]amino}pyrimidin-4-yl]amino}bicyclo[2.2.1]hept-5-ene-2-carboxamide
(1S,2S,3R,4R)-3-{[5-...
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1

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EBC-609086
EBC-609086

CAS:2764615-56-5

1,1-dioxo-N-{3-[4-(trifluoromethoxy)benzenesulfonamido]propyl}-1lambda6-benzothiophene-2-carboxamide
1,1-dioxo-N-{3-[4-(t...
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1

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