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Product details:
CAS
1616391-65-1
Purity
95%
EPZ015666 inhibits PRMT5 directly in cell-free experiments. This is a chemical probe with oral bioavailability and demonstrated efficacy in mouse xenograft models, both with reduction in tumor volume (Z-138 and Maver-1 cells) and PRMT5 target inhibition (SDMA levels).
Properties
Name
EPZ015666
Smiles
O[C@@H](CNC(=O)C=1C=C(NC2COC2)N=CN1)CN3CCC=4C=CC=CC4C3
Targets
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Target name
Target pX
Target action
doi
SDS
EPZ015666 | GSK3235025
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$127
2 mg
$132
5 mg
$144
10 mg
$159
15 mg
$225
20 mg
$290
25 mg
$359
30 mg
$405
35 mg
$451
40 mg
$492
45 mg
$541
50 mg
$582
75 mg
$851
100 mg
$POA
Quantity
1
Total amount
$ 144
EPZ015666 | GSK3235025
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.