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Product details:
CAS
1952247-05-0
Purity
95%
PD00017273 is an inhibitor of human PARG enzyme with IC50 of 12 nM and good selectivity over the two closest functional homologues, PARP1 and ARH3 (>100 μM). It is suitable for use in cellular assays and is not cytotoxic in HeLa cells up to 30 μM.
Properties
Name
PD00017273
Smiles
CC=1C=C(CN2C(=O)N(CC3=CN=C(C)S3)C(=O)C=4C=C(C=CC24)S(=O)(=O)NC5(C)CC5)N(C)N1
Targets
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Target name
Target pX
Target action
doi
SDS
PDD00017273
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$171
2 mg
$256
5 mg
$511
10 mg
$886
15 mg
$1073
20 mg
$1260
25 mg
$1533
30 mg
$1805
35 mg
$2078
40 mg
$2350
45 mg
$2520
50 mg
$2691
75 mg
$3576
100 mg
$POA
Quantity
1
Total amount
$ 511
PDD00017273
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.