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Product details:

GI254023X

Search by this structure
Molecule product

ID

EBC-516246

CAS

260264-93-5

Purity

95%

GI254023X is a selective inhibitor of ADAM10 with 100-fold selectivity for ADAM10 over ADAM17.

Properties

cLogP:2.492
MW:391.247

Name

GI254023X

Smiles

CNC(=O)[C@@H](NC(=O)[C@H](CCCC=1C=CC=CC1)[C@H](C)N(O)C=O)C(C)(C)C

Targets

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Chemical probes

Target name

Target pX

Target action

doi

Disintegrin and metalloproteinase domain-containing protein 10

7.57

Inhibitor

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Synonyms

GI254023X | SRI028594

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Prices

Temporarily unavailable

1 mg

$85

2 mg

$95

5 mg

$190

10 mg

$330

15 mg

$399

20 mg

$469

25 mg

$570

30 mg

$671

35 mg

$773

40 mg

$874

45 mg

$937

50 mg

$1000

75 mg

$1330

100 mg

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Quantity

-

1

+

Total amount

$ 190

Your current project

Temporarily unavailable

Synonyms

GI254023X | SRI028594

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Target activity features

It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.

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