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Product details:
CAS
2377335-74-3
Purity
95%
M-808 covalently reacts with C329 of Menin via its acrylamide moiety and thereby inhibits the Menin-MLL protein-protein interaction. It is a very potent and efficacious inhibitor in vitro and in cells.
Properties
Name
M-808
Smiles
COC(=O)N[C@H]1CCC[C@@H]1[C@@](CN2CCC2)(C3CCN(CC4CN(C4)C=5C=CC(=CC5)S(=O)(=O)C6CN(C6)C(=O)/C=C/CN7CCCCC7)CC3)C=8C=CC=C(F)C8
Targets
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Target name
Target pX
Target action
doi
SDS
No records
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$POA
2 mg
$POA
5 mg
$POA
10 mg
$POA
15 mg
$POA
20 mg
$POA
25 mg
$POA
30 mg
$POA
35 mg
$POA
40 mg
$POA
45 mg
$POA
50 mg
$POA
75 mg
$POA
100 mg
$POA
Quantity
1
Total amount
$ 0
No records
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.