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Product details:
CAS
1414797-35-5
Purity
95%
GSK2973980A is a potent and selective DGAT1 inhibitor (IC50 = 3 nM). GSK2973980A demonstrates excellent DMPK profiles and in vivo efficacy in a postprandial lipid excursion model in mice.
Properties
Name
GSK2973980A
Smiles
OC(=O)C[C@]1(CC(F)(F)F)CCC=2C=C(C=CC2C1=O)C=3C=NC(NC(=O)NC=4C=CC(F)=C(F)C4)=CN3
Targets
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Target name
Target pX
Target action
doi
SDS
GSK2973980A
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$POA
2 mg
$POA
5 mg
$POA
10 mg
$POA
15 mg
$POA
20 mg
$POA
25 mg
$POA
30 mg
$POA
35 mg
$POA
40 mg
$POA
45 mg
$POA
50 mg
$POA
75 mg
$POA
100 mg
$POA
Quantity
1
Total amount
$ 0
GSK2973980A
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.