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Product details:
ID
CAS
2519823-34-6
Purity
95%
BSJ-4-116 is a PROTAC connected by ligands for Cereblon and CDK. BSJ-4-116 is a highly potent and selective CDK12 degrader with an IC50 of 6 nM.
Properties
Name
BSJ-4-116
Smiles
CC(C)S(=O)(=O)C=1C=CC=CC1NC=2N=C(N[C@@H]3CCCN(CCCCCCCNC(=O)COC=4C=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C54)C3)N=CC2Cl
Targets
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Target name
Target pX
Target action
doi
BSJ-04-116
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$85
2 mg
$100
5 mg
$146
10 mg
$253
15 mg
$307
20 mg
$360
25 mg
$438
30 mg
$516
35 mg
$594
40 mg
$672
45 mg
$720
50 mg
$769
75 mg
$1022
100 mg
$POA
Quantity
1
Total amount
$ 146
BSJ-04-116
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.