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Product details:

GSK8612

Search by this structure
Molecule product

ID

EBC-157116

|

CAS

2361659-62-1

Purity

95%

GSK8612 is a highly selective and potent Tank-binding Kinase-1 inhibitor, with a pIC50 of 8.5 for recombinant TBK1.

Properties

cLogP:2.518
MW:520.327

Name

GSK8612

Smiles

CC1=NN(CC(F)(F)F)C=C1NC=2N=CC(Br)=C(NCC=3C=CC(=CC3)S(=O)(=O)N)N2

Targets

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Chemical probes

Target name

Target pX

Target action

doi

Serine/threonine-protein kinase TBK1

8.1

Inhibitor

Open link
Synonyms

GSK8612

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Prices

1 mg

$82

2 mg

$84

5 mg

$89

10 mg

$115

15 mg

$156

20 mg

$195

25 mg

$214

30 mg

$236

35 mg

$255

40 mg

$276

45 mg

$297

50 mg

$336

75 mg

$502

100 mg

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Quantity

-

1

+

Total amount

$ 89

Your current project

In Stock

Synonyms

GSK8612

Transportation & Handlings
Storage temperature:RT
Transport temperature:Standard
Dangerous goods:No
Solubility

No data available

Purity & Quality Control

The compound has purity validated by NMR and/or LCMS methods.

Target activity features

It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.

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Related Compounds

EBC-157116
EBC-157116

CAS:2361659-62-1

GSK8612
GSK8612
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0

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