Terfenadine

We provide 1 form of Terfenadine

Molecule smiles
Name

Terfenadine

Properties
CAS:

50679-08-8

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MW:

471.673

|

cLogP:

6.073

Description

Terfenadine is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistaminic and non-sedative effects. Terfenadine's active metabolite competitively binds peripheral H1-receptors, thereby stabilizing an inactive conformation of the receptor.

Synonyms

terfenadine | terfenedine

Description

Terfenadine is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist with antihistaminic and non-sedative effects. Terfenadine's active metabolite competitively binds peripheral H1-receptors, thereby stabilizing an inactive conformation of the receptor.

Synonyms

terfenadine | terfenedine

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1

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Temporarily unavailable

Impurities and Related Compounds

We provide 0 compound for Terfenadine