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Product details:
CAS
942206-85-1
Purity
95%
GSK1016790A is a highly potent agonist of TRPV4. The available data use complementary cell based assays to establish that human TRPV4 is activated with EC50 3-5 nM while mouse TRPV4 potency is somewhat lower, 18 nM.
Properties
Name
GSK1016790A
Smiles
CC(C)C[C@H](NC(=O)C1=CC=2C=CC=CC2S1)C(=O)N3CCN(CC3)C(=O)[C@H](CO)NS(=O)(=O)C=4C=CC(Cl)=CC4Cl
Targets
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Target name
Target pX
Target action
doi
SDS
GSK101 | GSK1016790A
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$121
2 mg
$127
5 mg
$138
10 mg
$153
15 mg
$216
20 mg
$278
25 mg
$345
30 mg
$389
35 mg
$433
40 mg
$472
45 mg
$520
50 mg
$558
75 mg
$816
100 mg
$POA
Quantity
1
Total amount
$ 138
GSK101 | GSK1016790A
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.