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Product details:
CAS
1338466-77-5
Purity
95%
EPZ004777 is a potent and selective DOT1L inhibitor with an IC50 of 0.4 nM.
Properties
Name
EPZ004777
Smiles
CC(C)N(CCCNC(=O)NC=1C=CC(=CC1)C(C)(C)C)C[C@H]2O[C@H]([C@H](O)[C@@H]2O)N3C=CC=4C(N)=NC=NC34
Targets
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Target name
Target pX
Target action
doi
EPZ-4777 | EPZ004777
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$102
2 mg
$103
5 mg
$111
10 mg
$122
15 mg
$171
20 mg
$219
25 mg
$280
30 mg
$320
35 mg
$353
40 mg
$394
45 mg
$435
50 mg
$483
75 mg
$624
100 mg
$POA
Quantity
1
Total amount
$ 111
EPZ-4777 | EPZ004777
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.