Compound libraries
Products
EBC main page
Search
Dyes
Impurities
Chemical probes
Contacts us
Pfizer reference compounds
Services
© 2026 Copyright Enamine
Back
Product details:
CAS
1337532-29-2
Purity
95%
GSK2656157 is a selective inhibitor of PERK kinase (EIF2AK3) that binds the nucleotide pocket. In terms of selectivity in binding potency, it is at least 500-fold selective over other members of the EIF2AK family, with minimal inhibition of other off kinases when surveyed in a broad panel (300 kinases).
Properties
Name
GSK2656157
Smiles
CC=1C=CC=C(CC(=O)N2CCC=3C2=CC=C(C4=CN(C)C=5N=CN=C(N)C45)C3F)N1
Targets
Please log in to see this information
Target name
Target pX
Target action
doi
GSK2656157
No data available
The compound has purity validated by NMR and/or LCMS methods.
1 mg
$75
2 mg
$77
5 mg
$82
10 mg
$107
15 mg
$144
20 mg
$180
25 mg
$197
30 mg
$217
35 mg
$235
40 mg
$254
45 mg
$274
50 mg
$309
75 mg
$462
100 mg
$POA
Quantity
1
Total amount
$ 82
GSK2656157
No data available
The compound has purity validated by NMR and/or LCMS methods.
Target activity features
It should be emphasized that the product may be active against a larger number of targets than shown on the card. The information represented here refers to the targets with the largest value of pX or the targets with ΔpX less than 1.5 from the largest pX value.