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Clinical trials play a vital role in the discovery of new medicines. They go through a series of phases to test whether a potential drug is safe and whether it works on humans. If the compound successively passes all phases of clinical trials, it can be submitted for FDA (or other pharmaceutical regulatory agency) approval to become a novel drug. Also, a drug with established effectiveness and bioactivity against one disease may be useful in discovering a new drug indication. The process of re-using known drugs to find a new cure for other diseases is called drug repurposing.
FDA Approved and Potential Drugs library is combined of FDA approved drugs, drug repurposing pharmaceuticals, and compounds that passed at least the first phase of clinical trials. It contains 1975 compounds. Additional information about the clinical trials phase and national clinical trial (NCT) numbers is also available to get a review of the clinical success of the substance.
Related terms: H1 receptor, D2 receptor, carbonic anhydrase, 5-HT2A receptor, acetylcholinesterase, COX-1, epidermal growth factor receptor, COX-2, D3 receptor
Remdesivir is a nucleoside analog used to treat RNA virus infections.
Zorifertinib is a potent, orally active, central nervous system-penetrant, EGFR inhibitor with IC50 = 0.5nM.
Tiapride is a selective D2 and D3 dopamine receptor blocker in the brain. Tiapride is indicated for the treatment of a variety of neurological and psychiatric disorders
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NoteAll the compounds with solubility below 10 mM are shipped as 2 mM solutions.
H1 receptor
45
45
Number of compounds
45
D2 receptor
40
40
Number of compounds
40
carbonic anhydrase 2
34
34
Number of compounds
34
5-HT2A receptor
33
33
Number of compounds
33
acetylcholinesterase (Cartwright blood group)
30
30
Number of compounds
30
COX-1
30
30
Number of compounds
30
epidermal growth factor receptor
29
29
Number of compounds
29
Kv11.1
27
27
Number of compounds
27
carbonic anhydrase 1
24
24
Number of compounds
24
carbonic anhydrase 9
23
23
Number of compounds
23
COX-2
21
21
Number of compounds
21
D3 receptor
21
21
Number of compounds
21
ABCB1
21
21
Number of compounds
21
M1 receptor
21
21
Number of compounds
21
CYP1A2
20
20
Number of compounds
20
Androgen receptor
20
20
Number of compounds
20
carbonic anhydrase 12
20
20
Number of compounds
20
β2-adrenoceptor
19
19
Number of compounds
19
SERT
17
17
Number of compounds
17
α1A-adrenoceptor
17
17
Number of compounds
17
M2 receptor
17
17
Number of compounds
17
Cav1.1
17
17
Number of compounds
17
CYP1A1
16
16
Number of compounds
16
ABCG2
15
15
Number of compounds
15
dihydrofolate reductase
15
15
Number of compounds
15
5-HT3A
14
14
Number of compounds
14
sigma non-opioid intracellular receptor 1
14
14
Number of compounds
14
Janus kinase 2
14
14
Number of compounds
14
β1-adrenoceptor
14
14
Number of compounds
14
α1B-adrenoceptor
13
13
Number of compounds
13
M3 receptor
13
13
Number of compounds
13
carbonic anhydrase 7
13
13
Number of compounds
13
serine protease 1
13
13
Number of compounds
13
erb-b2 receptor tyrosine kinase 2
13
13
Number of compounds
13
α2B-adrenoceptor
12
12
Number of compounds
12
5-HT2C receptor
12
12
Number of compounds
12
α2A-adrenoceptor
12
12
Number of compounds
12
Monoamine oxidase A
12
12
Number of compounds
12
amine oxidase copper containing 3
12
12
Number of compounds
12
D1 receptor
12
12
Number of compounds
12
fms related receptor tyrosine kinase 3
12
12
Number of compounds
12
Organic anion transporter 3
11
11
Number of compounds
11
A1 receptor
11
11
Number of compounds
11
5-HT1A receptor
11
11
Number of compounds
11
5-HT2B receptor
11
11
Number of compounds
11
Monoamine oxidase B
11
11
Number of compounds
11
Cav1.2
11
11
Number of compounds
11
CYP2E1
11
11
Number of compounds
11
TRPV1
11
11
Number of compounds
11
carbonic anhydrase 4
11
11
Number of compounds
11
histone deacetylase 1
10
10
Number of compounds
10
5-HT1B receptor
10
10
Number of compounds
10
Glucocorticoid receptor
10
10
Number of compounds
10
Janus kinase 3
10
10
Number of compounds
10
Aryl hydrocarbon receptor
10
10
Number of compounds
10
M4 receptor
10
10
Number of compounds
10
kinase insert domain receptor
10
10
Number of compounds
10
carbonic anhydrase 14
10
10
Number of compounds
10
butyrylcholinesterase
10
10
Number of compounds
10
tubulin alpha 1a
10
10
Number of compounds
10
Kv9.1
9
9
Number of compounds
9
5-HT6 receptor
9
9
Number of compounds
9
GABAA receptor α1 subunit
9
9
Number of compounds
9
Kir6.2
9
9
Number of compounds
9
Janus kinase 1
9
9
Number of compounds
9
Progesterone receptor
9
9
Number of compounds
9
Peroxisome proliferator-activated receptor-γ
9
9
Number of compounds
9
ATP-binding cassette, sub-family C (CFTR/MRP), member 8
8
8
Number of compounds
8
A2A receptor
8
8
Number of compounds
8
α1D-adrenoceptor
8
8
Number of compounds
8
α2C-adrenoceptor
8
8
Number of compounds
8
KNa1.1
8
8
Number of compounds
8
Organic cation transporter 1
8
8
Number of compounds
8
M5 receptor
8
8
Number of compounds
8
GABAA receptor β2 subunit
8
8
Number of compounds
8
GABAA receptor δ subunit
8
8
Number of compounds
8
5-HT1D receptor
8
8
Number of compounds
8
MDM2 proto-oncogene
8
8
Number of compounds
8
DAT
8
8
Number of compounds
8
platelet derived growth factor receptor alpha
8
8
Number of compounds
8
platelet derived growth factor receptor beta
8
8
Number of compounds
8
CoV 3C-like (main) protease
8
8
Number of compounds
8
sepiapterin reductase
8
8
Number of compounds
8
AT1 receptor
8
8
Number of compounds
8
cyclin dependent kinase 2
8
8
Number of compounds
8
Organic anion transporter 1
7
7
Number of compounds
7
5-LOX
7
7
Number of compounds
7
GluN2D
7
7
Number of compounds
7
A3 receptor
7
7
Number of compounds
7
H2 receptor
7
7
Number of compounds
7
Nav1.7
7
7
Number of compounds
7
5-HT7 receptor
7
7
Number of compounds
7
Mineralocorticoid receptor
7
7
Number of compounds
7
tyrosine kinase 2
7
7
Number of compounds
7
D4 receptor
7
7
Number of compounds
7
Peroxisome proliferator-activated receptor-α
7
7
Number of compounds
7
heat shock protein 90 beta family member 1
7
7
Number of compounds
7
dipeptidyl peptidase 4
7
7
Number of compounds
7
NET
7
7
Number of compounds
7
Pregnane X receptor
7
7
Number of compounds
7
AKT serine/threonine kinase 1
7
7
Number of compounds
7
ret proto-oncogene
7
7
Number of compounds
7
cyclin dependent kinase 9
7
7
Number of compounds
7
carbonic anhydrase 13
7
7
Number of compounds
7
OATP1B1
6
6
Number of compounds
6
CYP51A1
6
6
Number of compounds
6
histone deacetylase 3
6
6
Number of compounds
6
histone deacetylase 6
6
6
Number of compounds
6
Organic cation transporter 3
6
6
Number of compounds
6
TRPA1
6
6
Number of compounds
6
ABL proto-oncogene 1, non-receptor tyrosine kinase
6
6
Number of compounds
6
CFTR
6
6
Number of compounds
6
nicotinic acetylcholine receptor α4 subunit
6
6
Number of compounds
6
nicotinic acetylcholine receptor β2 subunit
6
6
Number of compounds
6
σ2
6
6
Number of compounds
6
GluN2C
6
6
Number of compounds
6
ALK receptor tyrosine kinase
6
6
Number of compounds
6
CYP19A1
6
6
Number of compounds
6
CCR5
6
6
Number of compounds
6
CXCR4
6
6
Number of compounds
6
Angiotensin-converting enzyme
6
6
Number of compounds
6
fms related receptor tyrosine kinase 1
6
6
Number of compounds
6
phosphodiesterase 5A
6
6
Number of compounds
6
fms related receptor tyrosine kinase 4
6
6
Number of compounds
6
Insulin receptor
6
6
Number of compounds
6
CB1 receptor
5
5
Number of compounds
5
OATP1B3
5
5
Number of compounds
5
histone deacetylase 2
5
5
Number of compounds
5
KCa1.1
5
5
Number of compounds
5
farnesyl diphosphate synthase
5
5
Number of compounds
5
signal transducer and activator of transcription 3
5
5
Number of compounds
5
Multidrug and toxin extrusion
5
5
Number of compounds
5
AKR1C3
5
5
Number of compounds
5
Estrogen receptor-β
5
5
Number of compounds
5
myeloperoxidase
5
5
Number of compounds
5
glycine receptor α1 subunit
5
5
Number of compounds
5
colony stimulating factor 1 receptor
5
5
Number of compounds
5
Organic cation transporter 2
5
5
Number of compounds
5
MC3 receptor
5
5
Number of compounds
5
topoisomerase (DNA) I mitochondrial
5
5
Number of compounds
5
Raf-1 proto-oncogene, serine/threonine kinase
5
5
Number of compounds
5
aurora kinase B
5
5
Number of compounds
5
B-Raf proto-oncogene, serine/threonine kinase
5
5
Number of compounds
5
Vesicular monoamine transporter 2
4
4
Number of compounds
4
mitogen-activated protein kinase 1
4
4
Number of compounds
4
TA1 receptor
4
4
Number of compounds
4
CXCR1
4
4
Number of compounds
4
epoxide hydrolase 2
4
4
Number of compounds
4
SMO
4
4
Number of compounds
4
hydroxymethylglutaryl-CoA reductase
4
4
Number of compounds
4
discoidin domain receptor tyrosine kinase 2
4
4
Number of compounds
4
Angiotensin-converting enzyme 2
4
4
Number of compounds
4
Nav1.5
4
4
Number of compounds
4
leukocyte receptor tyrosine kinase
4
4
Number of compounds
4
LCK proto-oncogene, Src family tyrosine kinase
4
4
Number of compounds
4
5-HT4 receptor
4
4
Number of compounds
4
Nav1.1
4
4
Number of compounds
4
cyclin dependent kinase 7
4
4
Number of compounds
4
pancreatic lipase
4
4
Number of compounds
4
Bruton tyrosine kinase
4
4
Number of compounds
4
DNA methyltransferase 1
4
4
Number of compounds
4
CD4
4
4
Number of compounds
4
beta-secretase 1
4
4
Number of compounds
4
β3-adrenoceptor
4
4
Number of compounds
4
Organic cation/carnitine transporter 2
4
4
Number of compounds
4
maternal embryonic leucine zipper kinase
4
4
Number of compounds
4
cyclin dependent kinase 1
4
4
Number of compounds
4
neurotrophic receptor tyrosine kinase 1
4
4
Number of compounds
4
neurotrophic receptor tyrosine kinase 3
4
4
Number of compounds
4
CDC like kinase 4
4
4
Number of compounds
4
cyclin G associated kinase
4
4
Number of compounds
4
xanthine dehydrogenase
4
4
Number of compounds
4
coagulation factor II, thrombin
4
4
Number of compounds
4
CDC like kinase 2
4
4
Number of compounds
4
MMP2
4
4
Number of compounds
4
nicotinic acetylcholine receptor α7 subunit
4
4
Number of compounds
4
SRC proto-oncogene, non-receptor tyrosine kinase
4
4
Number of compounds
4
Kv7.1
4
4
Number of compounds
4
aurora kinase A
4
4
Number of compounds
4
MET proto-oncogene, receptor tyrosine kinase
4
4
Number of compounds
4
Kir6.1
4
4
Number of compounds
4
μ receptor
4
4
Number of compounds
4
OATP1A2
4
4
Number of compounds
4
5-HT3B
4
4
Number of compounds
4
MT1 receptor
4
4
Number of compounds
4
P2X7
4
4
Number of compounds
4
Endothelial NOS
4
4
Number of compounds
4
Inducible NOS
4
4
Number of compounds
4
Neuronal NOS
4
4
Number of compounds
4
transthyretin
4
4
Number of compounds
4
CYP17A1
4
4
Number of compounds
4
CYP11B2
4
4
Number of compounds
4
Rho associated coiled-coil containing protein kinase 2
4
4
Number of compounds
4
GABAA receptor α2 subunit
4
4
Number of compounds
4
GABAA receptor β3 subunit
4
4
Number of compounds
4
GABAA receptor γ2 subunit
4
4
Number of compounds
4
CB2 receptor
3
3
Number of compounds
3
poly(ADP-ribose) polymerase 1
3
3
Number of compounds
3
Nav1.8
3
3
Number of compounds
3
CYP7B1
3
3
Number of compounds
3
histone deacetylase 5
3
3
Number of compounds
3
Nav1.2
3
3
Number of compounds
3
A2B receptor
3
3
Number of compounds
3
CCR2
3
3
Number of compounds
3
CYP11B1
3
3
Number of compounds
3
GABAA receptor α5 subunit
3
3
Number of compounds
3
Cav2.2
3
3
Number of compounds
3
p21 (RAC1) activated kinase 1
3
3
Number of compounds
3
polo like kinase 3
3
3
Number of compounds
3
Retinoic acid receptor-β
3
3
Number of compounds
3
CYP1B1
3
3
Number of compounds
3
mitogen-activated protein kinase 3
3
3
Number of compounds
3
casein kinase 2, alpha 1 polypeptide subunit
3
3
Number of compounds
3
V2 receptor
3
3
Number of compounds
3
discoidin domain receptor tyrosine kinase 1
3
3
Number of compounds
3
ZAK sterile alpha motif and leucine zipper containing kinase AZK
3
3
Number of compounds
3
polo like kinase 1
3
3
Number of compounds
3
polo like kinase 2
3
3
Number of compounds
3
c-ros oncogene 1, receptor tyrosine kinase
3
3
Number of compounds
3
LYN proto-oncogene, Src family tyrosine kinase
3
3
Number of compounds
3
protein tyrosine kinase 2
3
3
Number of compounds
3
spleen associated tyrosine kinase
3
3
Number of compounds
3
AXL receptor tyrosine kinase
3
3
Number of compounds
3
integrin, alpha M subunit (complement component 3 receptor 3 subunit)
3
3
Number of compounds
3
protein kinase A
3
3
Number of compounds
3
AKT serine/threonine kinase 3
3
3
Number of compounds
3
AKT serine/threonine kinase 2
3
3
Number of compounds
3
KCa3.1
3
3
Number of compounds
3
Catechol-O-methyltransferase
3
3
Number of compounds
3
GABAA receptor α3 subunit
3
3
Number of compounds
3
H-PGDS
3
3
Number of compounds
3
proteasome 20S subunit beta 5
3
3
Number of compounds
3
synaptic vesicle glycoprotein 2A
3
3
Number of compounds
3
CaS receptor
3
3
Number of compounds
3
GPRC6 receptor
3
3
Number of compounds
3
CYP27A1
3
3
Number of compounds
3
H3 receptor
3
3
Number of compounds
3
Estrogen-related receptor-γ
3
3
Number of compounds
3
Arginase I
3
3
Number of compounds
3
mitogen-activated protein kinase kinase 1
3
3
Number of compounds
3
CysLT1 receptor
3
3
Number of compounds
3
Thyroid hormone receptor-α
3
3
Number of compounds
3
YES proto-oncogene 1, Src family tyrosine kinase
3
3
Number of compounds
3
MT2 receptor
3
3
Number of compounds
3
AP2 associated kinase 1
3
3
Number of compounds
3
mitogen-activated protein kinase kinase kinase kinase 2
3
3
Number of compounds
3
mitogen-activated protein kinase 8
3
3
Number of compounds
3
mitogen-activated protein kinase 10
3
3
Number of compounds
3
cyclin dependent kinase 5
3
3
Number of compounds
3
Rho associated coiled-coil containing protein kinase 1
3
3
Number of compounds
3
squalene monooxygenase
3
3
Number of compounds
3
NLRP3
3
3
Number of compounds
3
erb-b2 receptor tyrosine kinase 4
3
3
Number of compounds
3
GPBA receptor
3
3
Number of compounds
3
coagulation factor X
3
3
Number of compounds
3
mitogen-activated protein kinase 14
3
3
Number of compounds
3
Sodium/glucose cotransporter 2
3
3
Number of compounds
3
FFA1 receptor
3
3
Number of compounds
3
Organic anion transporter 2
3
3
Number of compounds
3
phosphodiesterase 4B
3
3
Number of compounds
3
aurora kinase C
3
3
Number of compounds
3
carboxylesterase 1
3
3
Number of compounds
3
cyclin dependent kinase 4
3
3
Number of compounds
3
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma
3
3
Number of compounds
3
PAF receptor
2
2
Number of compounds
2
Pim-1 proto-oncogene, serine/threonine kinase
2
2
Number of compounds
2
ABCB11
2
2
Number of compounds
2
tankyrase
2
2
Number of compounds
2
Farnesoid X receptor
2
2
Number of compounds
2
Equilibrative nucleoside transporter 2
2
2
Number of compounds
2
Plasma membrane monoamine transporter
2
2
Number of compounds
2
P2Y12 receptor
2
2
Number of compounds
2
protein kinase, cAMP-dependent, catalytic, alpha subunit
2
2
Number of compounds
2
ribosomal protein S6 kinase B1
2
2
Number of compounds
2
aldehyde dehydrogenase 2 family member
2
2
Number of compounds
2
GABAB2
2
2
Number of compounds
2
GABAA receptor α4 subunit
2
2
Number of compounds
2
GABAA receptor β1 subunit
2
2
Number of compounds
2
serum/glucocorticoid regulated kinase family member 3
2
2
Number of compounds
2
5-ht1e receptor
2
2
Number of compounds
2
activin A receptor type 1
2
2
Number of compounds
2
bone morphogenetic protein receptor type IB
2
2
Number of compounds
2
MATE2
2
2
Number of compounds
2
TRPC5
2
2
Number of compounds
2
ABCC9
2
2
Number of compounds
2
FER tyrosine kinase
2
2
Number of compounds
2
tyrosinase
2
2
Number of compounds
2
integrin, alpha 4 subunit (antigen CD49D, alpha 4 subunit of VLA-4 receptor)
2
2
Number of compounds
2
Methionyl aminopeptidase 1
2
2
Number of compounds
2
Methionyl aminopeptidase 2
2
2
Number of compounds
2
GlyT1
2
2
Number of compounds
2
EPH receptor B1
2
2
Number of compounds
2
carbonic anhydrase 5A
2
2
Number of compounds
2
fatty acid binding protein 2
2
2
Number of compounds
2
steroid 5 alpha-reductase 2
2
2
Number of compounds
2
Equilibrative nucleoside transporter 1
2
2
Number of compounds
2
bromodomain containing 2
2
2
Number of compounds
2
bromodomain testis associated
2
2
Number of compounds
2
FP receptor
2
2
Number of compounds
2
nicotinic acetylcholine receptor β4 subunit
2
2
Number of compounds
2
LPA1 receptor
2
2
Number of compounds
2
KCa2.1
2
2
Number of compounds
2
Kv4.3
2
2
Number of compounds
2
MER proto-oncogene, tyrosine kinase
2
2
Number of compounds
2
L-Aromatic amino-acid decarboxylase
2
2
Number of compounds
2
AT2 receptor
2
2
Number of compounds
2
Neutral endopeptidase
2
2
Number of compounds
2
protein kinase C eta
2
2
Number of compounds
2
transforming growth factor beta receptor 1
2
2
Number of compounds
2
SRSF protein kinase 3
2
2
Number of compounds
2
histone deacetylase 8
2
2
Number of compounds
2
protein kinase C iota
2
2
Number of compounds
2
glutathione-disulfide reductase
2
2
Number of compounds
2
NK1 receptor
2
2
Number of compounds
2
Monocarboxylate transporter 1
2
2
Number of compounds
2
TRPM8
2
2
Number of compounds
2
ABCC1
2
2
Number of compounds
2
MAPK interacting serine/threonine kinase 1
2
2
Number of compounds
2
fibroblast growth factor receptor 3
2
2
Number of compounds
2
fyn related Src family tyrosine kinase
2
2
Number of compounds
2
FYN proto-oncogene, Src family tyrosine kinase
2
2
Number of compounds
2
GPR35
2
2
Number of compounds
2
GPR84
2
2
Number of compounds
2
BMP2 inducible kinase
2
2
Number of compounds
2
dual specificity tyrosine phosphorylation regulated kinase 1A
2
2
Number of compounds
2
dual specificity tyrosine phosphorylation regulated kinase 2
2
2
Number of compounds
2
TTK protein kinase
2
2
Number of compounds
2
mitogen-activated protein kinase 9
2
2
Number of compounds
2
Monoacylglycerol lipase
2
2
Number of compounds
2
nicotinic acetylcholine receptor α3 subunit
2
2
Number of compounds
2
DNA (cytosine-5-)-methyltransferase 3α
2
2
Number of compounds
2
glycogen synthase kinase 3 beta
2
2
Number of compounds
2
mitogen-activated protein kinase kinase kinase kinase 4
2
2
Number of compounds
2
protein kinase N2
2
2
Number of compounds
2
Nav1.4
2
2
Number of compounds
2
Alanine/serine/cysteine transporter 2
2
2
Number of compounds
2
ABCC4
2
2
Number of compounds
2
Haem oxygenase 1
2
2
Number of compounds
2
BLK proto-oncogene, Src family tyrosine kinase
2
2
Number of compounds
2
BMX non-receptor tyrosine kinase
2
2
Number of compounds
2
TXK tyrosine kinase
2
2
Number of compounds
2
TP receptor
2
2
Number of compounds
2
RAR-related orphan receptor-γ
2
2
Number of compounds
2
checkpoint kinase 1
2
2
Number of compounds
2
thyroid peroxidase
2
2
Number of compounds
2
doublecortin like kinase 3
2
2
Number of compounds
2
mitogen-activated protein kinase kinase kinase 8
2
2
Number of compounds
2
serine/threonine kinase 16
2
2
Number of compounds
2
GluN2B
2
2
Number of compounds
2
MMP7
2
2
Number of compounds
2
Retinoic acid receptor-γ
2
2
Number of compounds
2
FPR1
2
2
Number of compounds
2
TLR7
2
2
Number of compounds
2
S-Adenosylhomocysteine hydrolase
2
2
Number of compounds
2
Sodium/glucose cotransporter 1
2
2
Number of compounds
2
kallikrein related peptidase 7
2
2
Number of compounds
2
CYP11A1
2
2
Number of compounds
2
PAR1
2
2
Number of compounds
2
Translocator protein
2
2
Number of compounds
2
Kv3.1
2
2
Number of compounds
2
Folate hydrolase (prostate-specific membrane antigen) 1
2
2
Number of compounds
2
phosphodiesterase 4D
2
2
Number of compounds
2
indoleamine 2,3-dioxygenase 1
2
2
Number of compounds
2
mitogen-activated protein kinase kinase 5
2
2
Number of compounds
2
NUAK family kinase 1
2
2
Number of compounds
2
fibroblast growth factor receptor 2
2
2
Number of compounds
2
Retinoid X receptor-α
2
2
Number of compounds
2
MMP3
2
2
Number of compounds
2
MMP13
2
2
Number of compounds
2
κ receptor
2
2
Number of compounds
2
FFA2 receptor
2
2
Number of compounds
2
CDC like kinase 1
2
2
Number of compounds
2
EP2 receptor
2
2
Number of compounds
2
WEE1 G2 checkpoint kinase
2
2
Number of compounds
2
interleukin 1 receptor associated kinase 1
2
2
Number of compounds
2
MAPK interacting serine/threonine kinase 2
2
2
Number of compounds
2
receptor interacting serine/threonine kinase 1
2
2
Number of compounds
2
tec protein tyrosine kinase
2
2
Number of compounds
2
mitogen-activated protein kinase kinase kinase 3
2
2
Number of compounds
2
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta
2
2
Number of compounds
2
CDC like kinase 3
2
2
Number of compounds
2
neurotrophic receptor tyrosine kinase 2
2
2
Number of compounds
2
Endothelin-converting enzyme 1
1
1
Number of compounds
1
4-hydroxyphenylpyruvate dioxygenase
1
1
Number of compounds
1
AMP kinase
1
1
Number of compounds
1
Cav3.1
1
1
Number of compounds
1
Adenosine deaminase
1
1
Number of compounds
1
CYP8B1
1
1
Number of compounds
1
CYP21A2
1
1
Number of compounds
1
GPR55
1
1
Number of compounds
1
RyR1
1
1
Number of compounds
1
coagulation factor IX
1
1
Number of compounds
1
vitamin K epoxide reductase complex subunit 1
1
1
Number of compounds
1
TRPM7
1
1
Number of compounds
1
GABAA receptor γ1 subunit
1
1
Number of compounds
1
Cav2.1
1
1
Number of compounds
1
GAT1
1
1
Number of compounds
1
5-HT1F receptor
1
1
Number of compounds
1
phosphodiesterase 8A
1
1
Number of compounds
1
TLR4
1
1
Number of compounds
1
TRPC4
1
1
Number of compounds
1
TRPC6
1
1
Number of compounds
1
Dipeptidase 1
1
1
Number of compounds
1
G protein subunit alpha q
1
1
Number of compounds
1
C-terminal Src kinase
1
1
Number of compounds
1
MMP14
1
1
Number of compounds
1
CHT
1
1
Number of compounds
1
integrin, alpha 1 subunit
1
1
Number of compounds
1
integrin, alpha 2 subunit (CD49B, alpha 2 subunit of VLA-2 receptor)
1
1
Number of compounds
1
integrin, beta 3 subunit (platelet glycoprotein IIIa, antigen CD61)
1
1
Number of compounds
1
CoV Spike glycoprotein
1
1
Number of compounds
1
PROT
1
1
Number of compounds
1
phosphodiesterase 7A
1
1
Number of compounds
1
GABAB1
1
1
Number of compounds
1
heat shock protein family A (Hsp70) member 1A
1
1
Number of compounds
1
NTS1 receptor
1
1
Number of compounds
1
mGlu6 receptor
1
1
Number of compounds
1
Excitatory amino acid transporter 4
1
1
Number of compounds
1
Kv3.3
1
1
Number of compounds
1
Kv3.4
1
1
Number of compounds
1
checkpoint kinase 2
1
1
Number of compounds
1
ABCC5
1
1
Number of compounds
1
Proton-coupled folate transporter
1
1
Number of compounds
1
ribosomal protein S6 kinase A5
1
1
Number of compounds
1
ENaC α
1
1
Number of compounds
1
ENaC β
1
1
Number of compounds
1
ENaC γ
1
1
Number of compounds
1
Prolylcarboxypeptidase
1
1
Number of compounds
1
Dipeptidyl-peptidase 7
1
1
Number of compounds
1
nicotinic acetylcholine receptor α5 subunit
1
1
Number of compounds
1
5-HT3AB
1
1
Number of compounds
1
Vitamin D receptor
1
1
Number of compounds
1
integrin, alpha 5 subunit (fibronectin receptor, alpha polypeptide)
1
1
Number of compounds
1
integrin, beta 1 subunit (fibronectin receptor, beta polypeptide, antigen CD29 includes MDF2, MSK12)
1
1
Number of compounds
1
mPGES1
1
1
Number of compounds
1
PLA2-G5
1
1
Number of compounds
1
CoV Envelope protein
1
1
Number of compounds
1
mGlu1 receptor
1
1
Number of compounds
1
Cystine/glutamate transporter
1
1
Number of compounds
1
TYRO3 protein tyrosine kinase
1
1
Number of compounds
1
Dopamine beta-hydroxylase (dopamine beta-monooxygenase)
1
1
Number of compounds
1
L-Tyrosine hydroxylase
1
1
Number of compounds
1
glycine receptor β subunit
1
1
Number of compounds
1
L-PGDS
1
1
Number of compounds
1
proteasome 20S subunit beta 2
1
1
Number of compounds
1
Transforming growth factor β receptor
1
1
Number of compounds
1
ubiquitin specific peptidase 14
1
1
Number of compounds
1
Ras converting CAAX endopeptidase 1
1
1
Number of compounds
1
SRSF protein kinase 1
1
1
Number of compounds
1
lysine demethylase 4E
1
1
Number of compounds
1
TLR2
1
1
Number of compounds
1
histone deacetylase 10
1
1
Number of compounds
1
H4 receptor
1
1
Number of compounds
1
Interleukin-4 receptor subunit α
1
1
Number of compounds
1
Interleukin-6 receptor
1
1
Number of compounds
1
ATP4A
1
1
Number of compounds
1
fatty acid binding protein 5
1
1
Number of compounds
1
NADPH oxidase 1
1
1
Number of compounds
1
Monocarboxylate transporter 2
1
1
Number of compounds
1
nucleotide binding oligomerization domain containing 1
1
1
Number of compounds
1
L-Tryptophan hydroxylase 1
1
1
Number of compounds
1
L-Tryptophan hydroxylase 2
1
1
Number of compounds
1
ABCA1
1
1
Number of compounds
1
endoplasmic reticulum to nucleus signaling 1
1
1
Number of compounds
1
receptor interacting serine/threonine kinase 2
1
1
Number of compounds
1
calcium/calmodulin dependent protein kinase kinase 1
1
1
Number of compounds
1
calcium/calmodulin dependent protein kinase kinase 2
1
1
Number of compounds
1
serum/glucocorticoid regulated kinase 1
1
1
Number of compounds
1
tumor necrosis factor receptor 1
1
1
Number of compounds
1
phosphatidylinositol-4-phosphate 3-kinase catalytic subunit type 2 beta
1
1
Number of compounds
1
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta
1
1
Number of compounds
1
protein kinase, DNA-activated, catalytic subunit
1
1
Number of compounds
1
P2X4
1
1
Number of compounds
1
Urate anion exchanger 1
1
1
Number of compounds
1
IP3 kinase A
1
1
Number of compounds
1
Caspase 1
1
1
Number of compounds
1
Leukotriene A4 hydrolase
1
1
Number of compounds
1
GlyT2
1
1
Number of compounds
1
S1P1 receptor
1
1
Number of compounds
1
S1P5 receptor
1
1
Number of compounds
1
ABCA8
1
1
Number of compounds
1
fibroblast growth factor receptor 1
1
1
Number of compounds
1
EPH receptor A2
1
1
Number of compounds
1
EPH receptor A5
1
1
Number of compounds
1
EPH receptor A8
1
1
Number of compounds
1
Kv1.5
1
1
Number of compounds
1
hydroxysteroid 17-beta dehydrogenase 2
1
1
Number of compounds
1
phosphodiesterase 2A
1
1
Number of compounds
1
casein kinase 1 delta
1
1
Number of compounds
1
microtubule affinity regulating kinase 3
1
1
Number of compounds
1
glycogen synthase kinase 3 alpha
1
1
Number of compounds
1
NIMA related kinase 4
1
1
Number of compounds
1
legumain
1
1
Number of compounds
1
choline O-acetyltransferase
1
1
Number of compounds
1
cathepsin L
1
1
Number of compounds
1
lysyl oxidase like 2
1
1
Number of compounds
1
lanosterol synthase
1
1
Number of compounds
1
DNA topoisomerase I
1
1
Number of compounds
1
DNA topoisomerase II alpha
1
1
Number of compounds
1
Fatty acid amide hydrolase-2
1
1
Number of compounds
1
Y5 receptor
1
1
Number of compounds
1
Acetyl-CoA carboxylase 1
1
1
Number of compounds
1
Acetyl-CoA carboxylase 2
1
1
Number of compounds
1
GPR6
1
1
Number of compounds
1
lipase G, endothelial type
1
1
Number of compounds
1
Diacylglycerol lipase α
1
1
Number of compounds
1
Constitutive androstane receptor
1
1
Number of compounds
1
GnRH1 receptor
1
1
Number of compounds
1
ATR serine/threonine kinase
1
1
Number of compounds
1
RTP Type A
1
1
Number of compounds
1
RTP Type E
1
1
Number of compounds
1
RTP Type S
1
1
Number of compounds
1
Vesicular glutamate transporter 3
1
1
Number of compounds
1
GluA1
1
1
Number of compounds
1
GluA2
1
1
Number of compounds
1
GluA3
1
1
Number of compounds
1
nicotinic acetylcholine receptor α6 subunit
1
1
Number of compounds
1
TAS2R38
1
1
Number of compounds
1
death associated protein kinase 1
1
1
Number of compounds
1
death associated protein kinase 3
1
1
Number of compounds
1
5-HT5A receptor
1
1
Number of compounds
1
nicotinic acetylcholine receptor α9 subunit
1
1
Number of compounds
1
nicotinic acetylcholine receptor α10 subunit
1
1
Number of compounds
1
TRPM2
1
1
Number of compounds
1
ribosomal protein S6 kinase A3
1
1
Number of compounds
1
mitochondrial pyruvate carrier 1
1
1
Number of compounds
1
FPR2/ALX
1
1
Number of compounds
1
Ornithine decarboxylase
1
1
Number of compounds
1
TLR8
1
1
Number of compounds
1
Interferon-γ receptor
1
1
Number of compounds
1
FKBP prolyl isomerase 1A
1
1
Number of compounds
1
Adenosine kinase
1
1
Number of compounds
1
plasminogen activator, urokinase
1
1
Number of compounds
1
Ecto-5'-Nucleotidase
1
1
Number of compounds
1
V1A receptor
1
1
Number of compounds
1
Estrogen-related receptor-α
1
1
Number of compounds
1
Kv7.2
1
1
Number of compounds
1
Kv7.3
1
1
Number of compounds
1
Caspase 9
1
1
Number of compounds
1
CXCR2
1
1
Number of compounds
1
nicotinic acetylcholine receptor α1 subunit
1
1
Number of compounds
1
nicotinic acetylcholine receptor β1 subunit
1
1
Number of compounds
1
nicotinic acetylcholine receptor δ subunit
1
1
Number of compounds
1
nicotinic acetylcholine receptor ε subunit
1
1
Number of compounds
1
GLP-1 receptor
1
1
Number of compounds
1
tankyrase 2
1
1
Number of compounds
1
embryonic ectoderm development
1
1
Number of compounds
1
phosphodiesterase 3A
1
1
Number of compounds
1
succinate receptor
1
1
Number of compounds
1
Na+/dicarboxylate cotransporter 3
1
1
Number of compounds
1
ClC-2
1
1
Number of compounds
1
Fatty acid amide hydrolase
1
1
Number of compounds
1
Nav1.3
1
1
Number of compounds
1
retinol binding protein 1
1
1
Number of compounds
1
CYP27C1
1
1
Number of compounds
1
advanced glycosylation end-product specific receptor
1
1
Number of compounds
1
ADAM17
1
1
Number of compounds
1
calcium/calmodulin-dependent protein kinase II alpha subunit
1
1
Number of compounds
1
tryptophan 2,3-dioxygenase
1
1
Number of compounds
1
3-Mercaptopyruvate sulfurtransferase
1
1
Number of compounds
1
Sialin
1
1
Number of compounds
1
kallikrein B1
1
1
Number of compounds
1
plasminogen activator, tissue type
1
1
Number of compounds
1
Kv1.3
1
1
Number of compounds
1
Cx46
1
1
Number of compounds
1
F-type ATPase α subunit
1
1
Number of compounds
1
NPC1 like intracellular cholesterol transporter 1
1
1
Number of compounds
1
ETA receptor
1
1
Number of compounds
1
ETB receptor
1
1
Number of compounds
1
nuclear receptor coactivator 1
1
1
Number of compounds
1
GABAA receptor α6 subunit
1
1
Number of compounds
1
ClC-1
1
1
Number of compounds
1
inosine monophosphate dehydrogenase 1
1
1
Number of compounds
1
inosine monophosphate dehydrogenase 2
1
1
Number of compounds
1
mGlu2 receptor
1
1
Number of compounds
1
mGlu3 receptor
1
1
Number of compounds
1
Glucose transporter 1
1
1
Number of compounds
1
Peptide transporter 2
1
1
Number of compounds
1
Retinoic acid receptor-α
1
1
Number of compounds
1
K2P3.1
1
1
Number of compounds
1
MC4 receptor
1
1
Number of compounds
1
MC5 receptor
1
1
Number of compounds
1
Adipo1 receptor
1
1
Number of compounds
1
Adipo2 receptor
1
1
Number of compounds
1
ubiquitin specific peptidase 5
1
1
Number of compounds
1
fatty acid binding protein 7
1
1
Number of compounds
1
phosphodiesterase 11A
1
1
Number of compounds
1
protein arginine methyltransferase 5
1
1
Number of compounds
1
Thyroid hormone receptor-β
1
1
Number of compounds
1
cyclin dependent kinase 12
1
1
Number of compounds
1
cyclin dependent kinase 13
1
1
Number of compounds
1
oxoglutarate receptor
1
1
Number of compounds
1
protein kinase AMP-activated catalytic subunit alpha 2
1
1
Number of compounds
1
protein kinase AMP-activated non-catalytic subunit beta 1
1
1
Number of compounds
1
protein kinase AMP-activated non-catalytic subunit gamma 1
1
1
Number of compounds
1
PAS domain containing serine/threonine kinase
1
1
Number of compounds
1
Aminopeptidase N
1
1
Number of compounds
1
Arginyl aminopeptidase
1
1
Number of compounds
1
Leucine aminopeptidase 3
1
1
Number of compounds
1
E1A binding protein p300
1
1
Number of compounds
1
Organic cation/carnitine transporter 1
1
1
Number of compounds
1
sirtuin 1
1
1
Number of compounds
1
sirtuin 2
1
1
Number of compounds
1
zeta chain of T cell receptor associated protein kinase 70
1
1
Number of compounds
1
TRPV2
1
1
Number of compounds
1
CatSper1
1
1
Number of compounds
1
glutaminase
1
1
Number of compounds
1
phosphodiesterase 4A
1
1
Number of compounds
1
phosphodiesterase 4C
1
1
Number of compounds
1
phosphodiesterase 10A
1
1
Number of compounds
1
FFA3 receptor
1
1
Number of compounds
1
Tyrosine aminotransferase
1
1
Number of compounds
1
EPH receptor B6
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 19
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 4
1
1
Number of compounds
1
NIMA related kinase 3
1
1
Number of compounds
1
WEE2 oocyte meiosis inhibiting kinase
1
1
Number of compounds
1
glutaminyl-peptide cyclotransferase
1
1
Number of compounds
1
activin A receptor type 1B
1
1
Number of compounds
1
tyrosine kinase with immunoglobulin like and EGF like domains 1
1
1
Number of compounds
1
muscle associated receptor tyrosine kinase
1
1
Number of compounds
1
A-Raf proto-oncogene, serine/threonine kinase
1
1
Number of compounds
1
calcium/calmodulin dependent protein kinase ID
1
1
Number of compounds
1
calcium/calmodulin dependent protein kinase IG
1
1
Number of compounds
1
calcium/calmodulin dependent protein kinase IV
1
1
Number of compounds
1
cyclin dependent kinase like 2
1
1
Number of compounds
1
component of inhibitor of nuclear factor kappa B kinase complex
1
1
Number of compounds
1
casein kinase 1 epsilon
1
1
Number of compounds
1
doublecortin like kinase 1
1
1
Number of compounds
1
dual serine/threonine and tyrosine protein kinase
1
1
Number of compounds
1
dual specificity tyrosine phosphorylation regulated kinase 1B
1
1
Number of compounds
1
homeodomain interacting protein kinase 2
1
1
Number of compounds
1
homeodomain interacting protein kinase 3
1
1
Number of compounds
1
homeodomain interacting protein kinase 4
1
1
Number of compounds
1
inhibitor of nuclear factor kappa B kinase subunit beta
1
1
Number of compounds
1
leucine rich repeat kinase 2
1
1
Number of compounds
1
mitogen-activated protein kinase kinase 3
1
1
Number of compounds
1
mitogen-activated protein kinase kinase 4
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 10
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 11
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 12
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 2
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 7
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase 9
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase kinase 3
1
1
Number of compounds
1
mitogen-activated protein kinase kinase kinase kinase 5
1
1
Number of compounds
1
mitogen-activated protein kinase 7
1
1
Number of compounds
1
MAPK activated protein kinase 2
1
1
Number of compounds
1
MAPK activated protein kinase 3
1
1
Number of compounds
1
microtubule affinity regulating kinase 1
1
1
Number of compounds
1
microtubule affinity regulating kinase 4
1
1
Number of compounds
1
megakaryocyte-associated tyrosine kinase
1
1
Number of compounds
1
misshapen like kinase 1
1
1
Number of compounds
1
myosin light chain kinase 3
1
1
Number of compounds
1
myosin light chain kinase family member 4
1
1
Number of compounds
1
NIMA related kinase 11
1
1
Number of compounds
1
NIMA related kinase 2
1
1
Number of compounds
1
NIMA related kinase 6
1
1
Number of compounds
1
NIMA related kinase 7
1
1
Number of compounds
1
NUAK family, SNF1-like kinase, 2
1
1
Number of compounds
1
oxidative stress responsive kinase 1
1
1
Number of compounds
1
phosphatidylinositol-5-phosphate 4-kinase type 2 beta
1
1
Number of compounds
1
phosphatidylinositol-5-phosphate 4-kinase type 2 gamma
1
1
Number of compounds
1
phosphatidylinositol-4-phosphate 5-kinase type 1 alpha
1
1
Number of compounds
1
pre-mRNA processing factor 4B
1
1
Number of compounds
1
RIO kinase 1
1
1
Number of compounds
1
RIO kinase 3
1
1
Number of compounds
1
receptor interacting serine/threonine kinase 3
1
1
Number of compounds
1
STE20 like kinase
1
1
Number of compounds
1
src-related kinase lacking C-terminal regulatory tyrosine and N-terminal myristylation sites
1
1
Number of compounds
1
SRSF protein kinase 2
1
1
Number of compounds
1
serine/threonine kinase 11
1
1
Number of compounds
1
serine/threonine kinase 17b
1
1
Number of compounds
1
serine/threonine kinase 25
1
1
Number of compounds
1
serine/threonine kinase 3
1
1
Number of compounds
1
TAO kinase 1
1
1
Number of compounds
1
TAO kinase 3
1
1
Number of compounds
1
tau tubulin kinase 1
1
1
Number of compounds
1
tau tubulin kinase 2
1
1
Number of compounds
1
unc-51 like autophagy activating kinase 1
1
1
Number of compounds
1
unc-51 like autophagy activating kinase 2
1
1
Number of compounds
1
unc-51 like kinase 3
1
1
Number of compounds
1
VRK serine/threonine kinase 2
1
1
Number of compounds
1
WNK lysine deficient protein kinase 1
1
1
Number of compounds
1
WNK lysine deficient protein kinase 2
1
1
Number of compounds
1
beta adrenergic receptor kinase 1
1
1
Number of compounds
1
beta adrenergic receptor kinase 2
1
1
Number of compounds
1
G protein-coupled receptor kinase 4
1
1
Number of compounds
1
G protein-coupled receptor kinase 5
1
1
Number of compounds
1
protein kinase D1
1
1
Number of compounds
1
mitogen-activated protein kinase 11
1
1
Number of compounds
1
mitogen-activated protein kinase 12
1
1
Number of compounds
1
mitogen-activated protein kinase 13
1
1
Number of compounds
1
DM1 protein kinase
1
1
Number of compounds
1
citron rho-interacting serine/threonine kinase
1
1
Number of compounds
1
Serine/threonine kinase 38
1
1
Number of compounds
1
Serine/threonine kinase 38 like
1
1
Number of compounds
1
protein kinase N1
1
1
Number of compounds
1
ribosomal protein S6 kinase B2
1
1
Number of compounds
1
serine/threonine kinase 32B
1
1
Number of compounds
1
serine/threonine kinase 32C
1
1
Number of compounds
1
myosin light chain kinase 2
1
1
Number of compounds
1
P2X1
1
1
Number of compounds
1
P2X2
1
1
Number of compounds
1
P2X3
1
1
Number of compounds
1
Kir3.4
1
1
Number of compounds
1
DP1 receptor
1
1
Number of compounds
1
IP receptor
1
1
Number of compounds
1
mGlu5 receptor
1
1
Number of compounds
1
Rap guanine nucleotide exchange factor 3
1
1
Number of compounds
1
Rap guanine nucleotide exchange factor 4
1
1
Number of compounds
1
CaCC
1
1
Number of compounds
1
TRPM3
1
1
Number of compounds
1
15-LOX-1
1
1
Number of compounds
1
proteasome 20S subunit beta 1
1
1
Number of compounds
1
proteasome 20S subunit beta 8
1
1
Number of compounds
1
proteasome 20S subunit beta 9
1
1
Number of compounds
1
RyR2
1
1
Number of compounds
1
OATP2B1
1
1
Number of compounds
1
MMP12
1
1
Number of compounds
1
Sodium/calcium exchanger 1
1
1
Number of compounds
1
cyclin dependent kinase 6
1
1
Number of compounds
1
phosphatase and tensin homolog
1
1
Number of compounds
1
geranylgeranyl diphosphate synthase
1
1
Number of compounds
1
FGR proto-oncogene, Src family tyrosine kinase
1
1
Number of compounds
1
MMP9
1
1
Number of compounds
1
interleukin 1 receptor associated kinase 4
1
1
Number of compounds
1
renin
1
1
Number of compounds
1
V-type ATPase V1 motor A subunit
1
1
Number of compounds
1
nerve growth factor receptor
1
1
Number of compounds
1
3-phosphoinositide dependent protein kinase 1
1
1
Number of compounds
1
δ receptor
1
1
Number of compounds
1
cyclin dependent kinase 14
1
1
Number of compounds
1
cyclin dependent kinase 16
1
1
Number of compounds
1
cyclin dependent kinase 17
1
1
Number of compounds
1
activin A receptor type IL
1
1
Number of compounds
1
prolyl endopeptidase
1
1
Number of compounds
1
EPH receptor B2
1
1
Number of compounds
1
4-aminobutyrate aminotransferase
1
1
Number of compounds
1
NPFF1 receptor
1
1
Number of compounds
1
CoV Non-structural protein 8
1
1
Number of compounds
1
nuclear receptor coactivator 2
1
1
Number of compounds
1
PLCγ2
1
1
Number of compounds
1
ADAMTS4
1
1
Number of compounds
1
ADAMTS5
1
1
Number of compounds
1
TRH-specific aminopeptidase
1
1
Number of compounds
1
myosin light chain kinase
1
1
Number of compounds
1
mitogen-activated protein kinase 4
1
1
Number of compounds
1
B1 receptor
1
1
Number of compounds
1
B2 receptor
1
1
Number of compounds
1
Sodium/bile acid and sulphated solute cotransporter 2
1
1
Number of compounds
1
bromodomain and PHD finger containing 1
1
1
Number of compounds
1
motilin receptor
1
1
Number of compounds
1
MMP8
1
1
Number of compounds
1
EBCL-0028