Compound libraries
Products
EBC main page
Search
Impurities
Chemical probes
Contact
Services
© 2026 Copyright Enamine
Back
Protein kinases are enzymes that catalyze the transfer of phosphate groups from ATP molecules to various substrates. The process is known as phosphorylation. Kinases regulate many cellar functions, so the overaction of protein kinases in cancer cells may cause fast tumor growth. Thus, kinase-inhibiting molecules might act as antitumor agents and can be used in cancer treatments.
Kinase Inhibitor Library designed by our specialists contains 368 carefully selected small kinase inhibitors. It covers the wide scope of kinase targets and includes approved drugs, highly selective and broad-spectrum inhibitors, and the most recent discoveries.
Related terms: receptor tyrosine kinase, RTK, nRTK, CAMK, calcium/calmodulin-dependent protein kinase, mitogen-activated protein kinase, MAP, cyclin-dependent kinase, CDK, glycogen synthase kinase, GSK
Кinase action on substrate(Created by BioRender.com)
Fedratinib, approved 2019, cancer EBC-17140
Selective MAPK-14 inhibitor EBC-12783
H-7 is a broad spectrum kinase inhibitor EBC-101110
AAK1 and BMP2K inhibitor (2020) EBC-47126
We propose the complete list of Services powered by Enamine
All our products are for research purpose only. Any personal or non-scientific use is strictly prohibited.
NoteAll the compounds with solubility below 10 mM are shipped as 2 mM solutions.
Receptor tyrosine kinases (RTKs)
271
271
Number of compounds
271
Non-receptor tyrosine kinases (nRTKs)
146
146
Number of compounds
146
Mitogen-activated protein kinases (MAP kinases)
54
54
Number of compounds
54
CAMK: Calcium/calmodulin-dependent protein kinases
43
43
Number of compounds
43
Cyclin-dependent kinase (CDK) family
32
32
Number of compounds
32
Glycogen synthase kinase (GSK) family
30
30
Number of compounds
30
CMGC: Containing CDK, MAPK, GSK3, CLK families
29
29
Number of compounds
29
CAMK-like (CAMKL) family
27
27
Number of compounds
27
AGC: Containing PKA, PKG, PKC families
22
22
Number of compounds
22
STE20 family
22
22
Number of compounds
22
CK1: Casein kinase 1
22
22
Number of compounds
22
Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase (DYRK) family
22
22
Number of compounds
22
Casein kinase 2 (CK2) family
15
15
Number of compounds
15
Interleukin-1 receptor-associated kinase (IRAK) family
15
15
Number of compounds
15
Protein kinase C (PKC) family
14
14
Number of compounds
14
STE: Homologs of yeast Sterile 7, Sterile 11, Sterile 20 kinases
14
14
Number of compounds
14
Aurora kinase (Aur) family
13
13
Number of compounds
13
RSK family
12
12
Number of compounds
12
DMPK family
12
12
Number of compounds
12
Glycerophospholipid turnover
12
12
Number of compounds
12
RAF family
12
12
Number of compounds
12
IKK family
11
11
Number of compounds
11
Polo-like kinase (PLK) family
10
10
Number of compounds
10
Receptor serine/threonine kinase (RSTK) family
9
9
Number of compounds
9
Leucine-rich repeat kinase (LRRK) family
8
8
Number of compounds
8
LIM domain kinase (LISK) family
7
7
Number of compounds
7
G protein-coupled receptor kinases (GRKs)
6
6
Number of compounds
6
Phosphatidyl inositol 3' kinase-related kinases (PIKK) family
6
6
Number of compounds
6
NIMA (never in mitosis gene a)- related kinase (NEK) family
5
5
Number of compounds
5
WEE family
5
5
Number of compounds
5
Numb-associated kinase (NAK) family
5
5
Number of compounds
5
Mixed Lineage Kinase (MLK) family
4
4
Number of compounds
4
MAPK-Activated Protein Kinase (MAPKAPK) family
4
4
Number of compounds
4
IRE family
4
4
Number of compounds
4
NAK family
4
4
Number of compounds
4
Receptor interacting protein kinase (RIPK) family
4
4
Number of compounds
4
Lipid modifying kinases
3
3
Number of compounds
3
RIO family
2
2
Number of compounds
2
TKL-unique family
2
2
Number of compounds
2
Haspin family
1
1
Number of compounds
1
CAMKK family
1
1
Number of compounds
1
Inositol phosphate turnover
1
1
Number of compounds
1
Alpha kinase family
1
1
Number of compounds
1
TTK family
1
1
Number of compounds
1
Unc-51-like kinase (ULK) family
1
1
Number of compounds
1
EBCL-0020