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Transporters or membrane transport proteins assist in the movement of ions, small molecules, lipids, and macromolecules across biological membranes. Membrane transporters can be classified as ABC transporters (primary active transporters), P-type ATPases (transport enzymes that use the energy of hydrolysis to move ions across membranes), and the solute carrier family of transporters (SLCs, which act by secondary active transport and facilitative diffusion). Some diseases involve defects in the work of membrane transporters making them an important group of drug targets. For instance, ABC transporters play an essential role in the study of multi-drug resistance in cancer cells because of their ability to remove chemotherapeutic agents from the cell faster than they can cross the membrane. Inhibitors of the SLC family of transporters can be efficient in the treatment of many disorders, particularly depression (SERT), epilepsy (GABA transporter), and Parkinson's disease (DAT).
Transporter Ligands Library is composed of 799 small molecules.
Related terms: SERT, ABCG2, ABCB1, NET, ferroportin, DAT, organic anion transporter, organic cation transporter, ATP-binding cassette, CFTR/MRP, glucose transporter
Action of kinase transporter proteins(Created by BioRender.com)
Paroxetine is a serotinin reuptake inhibitor EBC-12122
VU046327 is a solute carrier family 12 member 5 inhibitor EBC-09061
ML-352 is a choline transporter 1 inhibitor EBC-12374
AR-C155858 is a MCT1 and MCT2 inhibitor EBC-46248
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NoteAll the compounds with solubility below 10 mM are shipped as 2 mM solutions.
SERT
36
36
Number of compounds
36
ABCG2
17
17
Number of compounds
17
ABCB1
17
17
Number of compounds
17
NET
17
17
Number of compounds
17
Ferroportin
14
14
Number of compounds
14
DAT
14
14
Number of compounds
14
Organic anion transporter 3
7
7
Number of compounds
7
Organic cation transporter 1
7
7
Number of compounds
7
Organic cation transporter 3
6
6
Number of compounds
6
Organic anion transporter 1
5
5
Number of compounds
5
Vesicular monoamine transporter 2
5
5
Number of compounds
5
Organic cation transporter 2
4
4
Number of compounds
4
Organic cation/carnitine transporter 2
4
4
Number of compounds
4
ATP-binding cassette, sub-family C (CFTR/MRP), member 8
4
4
Number of compounds
4
Glucose transporter 1
3
3
Number of compounds
3
GlyT1
3
3
Number of compounds
3
OATP1B3
3
3
Number of compounds
3
GlyT2
3
3
Number of compounds
3
Equilibrative nucleoside transporter 2
3
3
Number of compounds
3
Excitatory amino acid transporter 4
2
2
Number of compounds
2
Multidrug and toxin extrusion
2
2
Number of compounds
2
F-type ATPase α subunit
2
2
Number of compounds
2
CHT
2
2
Number of compounds
2
synaptic vesicle glycoprotein 2A
2
2
Number of compounds
2
Monocarboxylate transporter 1
2
2
Number of compounds
2
Fatty acid transport protein 1
2
2
Number of compounds
2
Urate anion exchanger 1
2
2
Number of compounds
2
OATP1B1
2
2
Number of compounds
2
Sodium/glucose cotransporter 2
2
2
Number of compounds
2
ABCC9
2
2
Number of compounds
2
SERCA1
2
2
Number of compounds
2
Na+/citrate cotransporter
2
2
Number of compounds
2
ABCB11
1
1
Number of compounds
1
V-type ATPase V1 motor A subunit
1
1
Number of compounds
1
Glucose transporter 4
1
1
Number of compounds
1
Alanine/serine/cysteine transporter 2
1
1
Number of compounds
1
ABCC5
1
1
Number of compounds
1
Proton-coupled folate transporter
1
1
Number of compounds
1
OATP1A2
1
1
Number of compounds
1
NPC intracellular cholesterol transporter 1
1
1
Number of compounds
1
Monocarboxylate transporter 4
1
1
Number of compounds
1
Monocarboxylate transporter 2
1
1
Number of compounds
1
GAT1
1
1
Number of compounds
1
Peptide transporter 2
1
1
Number of compounds
1
K-Cl cotransporter 2
1
1
Number of compounds
1
Sodium/glucose cotransporter 1
1
1
Number of compounds
1
DMT1
1
1
Number of compounds
1
Sodium/phosphate cotransporter 3
1
1
Number of compounds
1
Sodium-dependent phosphate transporter 1
1
1
Number of compounds
1
Sodium-dependent phosphate transporter 2
1
1
Number of compounds
1
Sodium phosphate 1
1
1
Number of compounds
1
ABCC1
1
1
Number of compounds
1
Plasma membrane monoamine transporter
1
1
Number of compounds
1
OATP2B1
1
1
Number of compounds
1
Excitatory amino acid transporter 1
1
1
Number of compounds
1
Excitatory amino acid transporter 2
1
1
Number of compounds
1
Sodium/nucleoside cotransporter 2
1
1
Number of compounds
1
Organic cation/carnitine transporter 1
1
1
Number of compounds
1
Vesicular acetylcholine transporter
1
1
Number of compounds
1
Glucose transporter 3
1
1
Number of compounds
1
Organic anion transporter 2
1
1
Number of compounds
1
Sodium/bile acid and sulphated solute cotransporter 2
1
1
Number of compounds
1
Equilibrative nucleoside transporter 1
1
1
Number of compounds
1
ATP4A
1
1
Number of compounds
1
EBCL-0023